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AZD7325

Glpbio
Catalog No:GC39342-10mM (in 1mL DMSO) CAS No.:942437-37-8 MDLNo: Brand:Glpbio purity: 特性: Purpose:AZD7325 是具有口服活性的 α2,3 receptor 的正向別構(gòu)調(diào)節(jié)劑 (PAM),Ki 分別是 0.3 and 1.3 nM,但在 α1 和 α5 受體亞型上效果較差。AZD7325 是一種中等 CYP1A2 和強(qiáng)效 CYP3A4 誘導(dǎo)劑。AZD7325 具有用于焦慮和 dravet 綜合征相關(guān)研究的潛力。DMSO: 250 mg/mL (705.46 mM)
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